PUBLICACIÓN

Glycosidase inhibition by all 10 stereoisomeric 2,5-dideoxy-2,5- iminohexitols prepared from the enantiomers of glucuronolactone

ACCEDER A LA PUBLICACIÓN: Scopus Orcid

Ayers B.J., Ngo N., Jenkinson S.F., Martinez R.F., Shimada Y., Adachi I., Weymouth-Wilson A.C., Kato A., Fleet G.W.J.

2012 JOURNAL OF ORGANIC CHEMISTRY

Organic Chemistry (Q1)

JCR: 4.564

SJR: 2.286

CITAS

39

DOI

10.1021/jo301243s

EID

2-s2.0-84868139436

ISSN

0022-3263

EISSN

1520-6904

BIBTEX

@article{Ayers_2012, doi = {10.1021/jo301243s}, url = {https://doi.org/10.1021%2Fjo301243s}, year = 2012, month = {sep}, publisher = {American Chemical Society ({ACS})}, volume = {77}, number = {18}, pages = {7777--7792}, author = {Benjamin J. Ayers and Nigel Ngo and Sarah F. Jenkinson and R. Fernando Mart{\'{\i}}nez and Yousuke Shimada and Isao Adachi and Alexander C. Weymouth-Wilson and Atsushi Kato and George W. J. Fleet}, title = {Glycosidase Inhibition by All 10 Stereoisomeric 2,5-Dideoxy-2,5-iminohexitols Prepared from the Enantiomers of Glucuronolactone}, journal = {The Journal of Organic Chemistry}}

AUTORES DE LA UEX

Rafael Fernando Martínez Vázquez

OTRAS PUBLICACIONES DE INTERÉS

An Efficient And Highly Diastereoselective Synthesis Of C-Glycosylated 1,3-Oxazolidines From N-Methyl-D-Glucamine
Catalytic Screening For 1,2-Diol Protection: A Saccharose-Derived Hydrothermal Carbon Showcases Enhanced Performance
Novel Graphitic Oxynitrides As Photocatalysts For Sustainable H2 Production And Co2 Valorization. The Importance Of Self-Assembly For Catalytic Activity
Catalytic Screening For 1,2-Diol Protection: A Saccharose-Derived Hydrothermal Carbon Showcases Enhanced Performance
Novel Graphitic Oxynitrides As Photocatalysts For Sustainable H2 Production And Co2 Valorization. The Importance Of Self-Assembly For Catalytic Activity
Tuning Synthesis And Sonochemistry Forges Learning And Enhances Educational Training: Protection Of 1,3-Diols Under Heterogeneous Catalysis As Sustainable Case Study
Novel Graphitic Oxynitrides As Photocatalysts For Sustainable H2 Production And Co2 Valorization. The Importance Of Self-Assembly For Catalytic Activity
Tuning Synthesis And Sonochemistry Forges Learning And Enhances Educational Training: Protection Of 1,3-Diols Under Heterogeneous Catalysis As Sustainable Case Study
Síntesis De Acetales Derivados De 1,2-Dioles En Presencia De Catalizadores Ácidos Carbonosos
Tuning Synthesis And Sonochemistry Forges Learning And Enhances Educational Training: Protection Of 1,3-Diols Under Heterogeneous Catalysis As Sustainable Case Study
Síntesis De Acetales Derivados De 1,2-Dioles En Presencia De Catalizadores Ácidos Carbonosos
A True Reverse Anomeric Effect Does Exist After All: A Hydrogen Bonding Stereocontrolling Effect In 2-Iminoaldoses
Síntesis De Acetales Derivados De 1,2-Dioles En Presencia De Catalizadores Ácidos Carbonosos
A True Reverse Anomeric Effect Does Exist After All: A Hydrogen Bonding Stereocontrolling Effect In 2-Iminoaldoses
University Students’ Introduction To Science Communication
A True Reverse Anomeric Effect Does Exist After All: A Hydrogen Bonding Stereocontrolling Effect In 2-Iminoaldoses
University Students’ Introduction To Science Communication
¿sabe El Estudiantado Universitario Hablar En Público?
University Students’ Introduction To Science Communication
¿sabe El Estudiantado Universitario Hablar En Público?
Preparación De Carbamatos A Partir De Aminas Aromáticas Mediante Catálisis Heterogénea
¿sabe El Estudiantado Universitario Hablar En Público?
Preparación De Carbamatos A Partir De Aminas Aromáticas Mediante Catálisis Heterogénea
An Eco-Friendly And Switchable Carbon-Based Catalyst For Protection-Deprotection Of Vicinal Diols
Preparación De Carbamatos A Partir De Aminas Aromáticas Mediante Catálisis Heterogénea
An Eco-Friendly And Switchable Carbon-Based Catalyst For Protection-Deprotection Of Vicinal Diols
Developing Public Speaking Skills In European Education Area Students: Reflections From Seven Years Of Experience
An Eco-Friendly And Switchable Carbon-Based Catalyst For Protection-Deprotection Of Vicinal Diols
Developing Public Speaking Skills In European Education Area Students: Reflections From Seven Years Of Experience
Mechanistic Insights Into The Oxidative Degradation Of Formic And Oxalic Acids With Ozone And Oh Radical. A Computational Rationale
Developing Public Speaking Skills In European Education Area Students: Reflections From Seven Years Of Experience
Mechanistic Insights Into The Oxidative Degradation Of Formic And Oxalic Acids With Ozone And Oh Radical. A Computational Rationale
Novel Antagonist Of The Type 2 Lysophosphatidic Acid Receptor (Lpa2), Ucm-14216, Ameliorates Spinal Cord Injury In Mice
Mechanistic Insights Into The Oxidative Degradation Of Formic And Oxalic Acids With Ozone And Oh Radical. A Computational Rationale
Novel Antagonist Of The Type 2 Lysophosphatidic Acid Receptor (Lpa2), Ucm-14216, Ameliorates Spinal Cord Injury In Mice
On The Origin Of Sugar Handedness: Facts, Hypotheses And Missing Links-A Review
Novel Antagonist Of The Type 2 Lysophosphatidic Acid Receptor (Lpa2), Ucm-14216, Ameliorates Spinal Cord Injury In Mice
On The Origin Of Sugar Handedness: Facts, Hypotheses And Missing Links-A Review
Discovery And Mechanism Of Action Studies Of 4,6-Diphenylpyrimidine-2-Carbohydrazides As Utrophin Modulators For The Treatment Of Duchenne Muscular Dystrophy
On The Origin Of Sugar Handedness: Facts, Hypotheses And Missing Links-A Review
Discovery And Mechanism Of Action Studies Of 4,6-Diphenylpyrimidine-2-Carbohydrazides As Utrophin Modulators For The Treatment Of Duchenne Muscular Dystrophy
Targeting The Ftsz Allosteric Binding Site With A Novel Fluorescence Polarization Screen, Cytological And Structural Approaches For Antibacterial Discovery
Discovery And Mechanism Of Action Studies Of 4,6-Diphenylpyrimidine-2-Carbohydrazides As Utrophin Modulators For The Treatment Of Duchenne Muscular Dystrophy
Targeting The Ftsz Allosteric Binding Site With A Novel Fluorescence Polarization Screen, Cytological And Structural Approaches For Antibacterial Discovery
Organic Sonochemistry: A Chemist's Timely Perspective On Mechanisms And Reactivity
Targeting The Ftsz Allosteric Binding Site With A Novel Fluorescence Polarization Screen, Cytological And Structural Approaches For Antibacterial Discovery
Organic Sonochemistry: A Chemist's Timely Perspective On Mechanisms And Reactivity
A Novel Agonist Of The Type 1 Lysophosphatidic Acid Receptor (Lpa1), Ucm-05194, Shows Efficacy In Neuropathic Pain Amelioration
Organic Sonochemistry: A Chemist's Timely Perspective On Mechanisms And Reactivity
A Novel Agonist Of The Type 1 Lysophosphatidic Acid Receptor (Lpa1), Ucm-05194, Shows Efficacy In Neuropathic Pain Amelioration
Imine Or Enamine? Insights And Predictive Guidelines From The Electronic Effect Of Substituents In H-Bonded Salicylimines
A Novel Agonist Of The Type 1 Lysophosphatidic Acid Receptor (Lpa1), Ucm-05194, Shows Efficacy In Neuropathic Pain Amelioration
Imine Or Enamine? Insights And Predictive Guidelines From The Electronic Effect Of Substituents In H-Bonded Salicylimines
Mutarotation Of Aldoses: Getting A Deeper Knowledge Of A Classic Equilibrium Enabled By Computational Analyses
Imine Or Enamine? Insights And Predictive Guidelines From The Electronic Effect Of Substituents In H-Bonded Salicylimines
Mutarotation Of Aldoses: Getting A Deeper Knowledge Of A Classic Equilibrium Enabled By Computational Analyses
A Novel Agonist Of The Type 1 Lysophosphatidic Acid Receptor (Lpa1), Ucm-05194, Shows Efficacy In Neuropathic Pain Amelioration.
Mutarotation Of Aldoses: Getting A Deeper Knowledge Of A Classic Equilibrium Enabled By Computational Analyses
A Novel Agonist Of The Type 1 Lysophosphatidic Acid Receptor (Lpa1), Ucm-05194, Shows Efficacy In Neuropathic Pain Amelioration.
Isolation From Stevia Rebaudiana Of Dmdp Acetic Acid, A Novel Iminosugar Amino Acid: Synthesis And Glycosidase Inhibition Profile Of Glycine And Β-Alanine Pyrrolidine Amino Acids
A Novel Agonist Of The Type 1 Lysophosphatidic Acid Receptor (Lpa1), Ucm-05194, Shows Efficacy In Neuropathic Pain Amelioration.
Isolation From Stevia Rebaudiana Of Dmdp Acetic Acid, A Novel Iminosugar Amino Acid: Synthesis And Glycosidase Inhibition Profile Of Glycine And Β-Alanine Pyrrolidine Amino Acids
Cycloadditions With Mesoionic Dipoles: Strategy And Control
Isolation From Stevia Rebaudiana Of Dmdp Acetic Acid, A Novel Iminosugar Amino Acid: Synthesis And Glycosidase Inhibition Profile Of Glycine And Β-Alanine Pyrrolidine Amino Acids
Cycloadditions With Mesoionic Dipoles: Strategy And Control
The Dimroth Rearrangement As A Probable Cause For Structural Misassignments In Imidazo[1,2-A]pyrimidines: A 15n-Labelling Study And An Easy Method For The Determination Of Regiochemistry
Cycloadditions With Mesoionic Dipoles: Strategy And Control
The Dimroth Rearrangement As A Probable Cause For Structural Misassignments In Imidazo[1,2-A]pyrimidines: A 15n-Labelling Study And An Easy Method For The Determination Of Regiochemistry
The Structural Assembly Switch Of Cell Division Protein Ftsz Probed With Fluorescent Allosteric Inhibitors
The Dimroth Rearrangement As A Probable Cause For Structural Misassignments In Imidazo[1,2-A]pyrimidines: A 15n-Labelling Study And An Easy Method For The Determination Of Regiochemistry
The Structural Assembly Switch Of Cell Division Protein Ftsz Probed With Fluorescent Allosteric Inhibitors
Cycloadditions With Mesoionic Dipoles: Strategy And Control
The Structural Assembly Switch Of Cell Division Protein Ftsz Probed With Fluorescent Allosteric Inhibitors
Cycloadditions With Mesoionic Dipoles: Strategy And Control
Structural Essentials For Β-: N -Acetylhexosaminidase Inhibition By Amides Of Prolines, Pipecolic And Azetidine Carboxylic Acids
Cycloadditions With Mesoionic Dipoles: Strategy And Control
Structural Essentials For Β-: N -Acetylhexosaminidase Inhibition By Amides Of Prolines, Pipecolic And Azetidine Carboxylic Acids
Nine Of 16 Stereoisomeric Polyhydroxylated Proline Amides Are Potent Β-N-Acetylhexosaminidase Inhibitors
Structural Essentials For Β-: N -Acetylhexosaminidase Inhibition By Amides Of Prolines, Pipecolic And Azetidine Carboxylic Acids
Nine Of 16 Stereoisomeric Polyhydroxylated Proline Amides Are Potent Β-N-Acetylhexosaminidase Inhibitors
Carbohydrate Derived Bicyclic Azetidin-3-Ones As Scaffolds For Highly Functionalized Azetidines
Nine Of 16 Stereoisomeric Polyhydroxylated Proline Amides Are Potent Β-N-Acetylhexosaminidase Inhibitors
Carbohydrate Derived Bicyclic Azetidin-3-Ones As Scaffolds For Highly Functionalized Azetidines
Short And Sweet: D-Glucose To L-Glucose And L-Glucuronic Acid
Carbohydrate Derived Bicyclic Azetidin-3-Ones As Scaffolds For Highly Functionalized Azetidines
Short And Sweet: D-Glucose To L-Glucose And L-Glucuronic Acid
Synthesis Of The Enantiomers Of Xylnac And Lyxnac: Comparison Of Β-N-Acetylhexosaminidase Inhibition By The 8 Stereoisomers Of 2-N-Acetylamino-1,2,4-Trideoxy-1,4-Iminopentitols
Short And Sweet: D-Glucose To L-Glucose And L-Glucuronic Acid
Synthesis Of The Enantiomers Of Xylnac And Lyxnac: Comparison Of Β-N-Acetylhexosaminidase Inhibition By The 8 Stereoisomers Of 2-N-Acetylamino-1,2,4-Trideoxy-1,4-Iminopentitols
Kurz Und Knapp:l-Glucose Undl-Glucuronsäure Ausd-Glucose
Synthesis Of The Enantiomers Of Xylnac And Lyxnac: Comparison Of Β-N-Acetylhexosaminidase Inhibition By The 8 Stereoisomers Of 2-N-Acetylamino-1,2,4-Trideoxy-1,4-Iminopentitols
Kurz Und Knapp:l-Glucose Undl-Glucuronsäure Ausd-Glucose
Hydrazones From Hydroxy Naphthaldehydes. Part 2. Condensations With Aromatic N-Aminoheterocycles And Elucidation Of Tautomeric Structures
Kurz Und Knapp:l-Glucose Undl-Glucuronsäure Ausd-Glucose
Hydrazones From Hydroxy Naphthaldehydes. Part 2. Condensations With Aromatic N-Aminoheterocycles And Elucidation Of Tautomeric Structures
(3r,4s,5r,6r,7s)-3,4,5,7-Tetrahydroxyconidine, An Azetidine Analogue Of 6,7-Diepicastanospermine And A Conformationally Constrained D- Deoxyaltronojirimycin, From L-Arabinose
Hydrazones From Hydroxy Naphthaldehydes. Part 2. Condensations With Aromatic N-Aminoheterocycles And Elucidation Of Tautomeric Structures
(3r,4s,5r,6r,7s)-3,4,5,7-Tetrahydroxyconidine, An Azetidine Analogue Of 6,7-Diepicastanospermine And A Conformationally Constrained D- Deoxyaltronojirimycin, From L-Arabinose
C-Branched Iminosugars: Α-Glucosidase Inhibition By Enantiomers Of Isodmdp, Isodgdp, And Isodab- L -Isodmdp Compared To Miglitol And Miglustat
(3r,4s,5r,6r,7s)-3,4,5,7-Tetrahydroxyconidine, An Azetidine Analogue Of 6,7-Diepicastanospermine And A Conformationally Constrained D- Deoxyaltronojirimycin, From L-Arabinose
C-Branched Iminosugars: Α-Glucosidase Inhibition By Enantiomers Of Isodmdp, Isodgdp, And Isodab- L -Isodmdp Compared To Miglitol And Miglustat
Azetidine Iminosugars From The Cyclization Of 3,5-Di- O -Triflates Of Α-Furanosides And Of 2,4-Di- O -Triflates Of Β-Pyranosides Derived From Glucose
C-Branched Iminosugars: Α-Glucosidase Inhibition By Enantiomers Of Isodmdp, Isodgdp, And Isodab- L -Isodmdp Compared To Miglitol And Miglustat
Azetidine Iminosugars From The Cyclization Of 3,5-Di- O -Triflates Of Α-Furanosides And Of 2,4-Di- O -Triflates Of Β-Pyranosides Derived From Glucose
N-(2-Carboxyethyl)-2,5-Dideoxy-2,5-Imino-D-Mannonic Acid [(3r,4r,5r)-1-(2-Carboxyethyl)-3,4-Dihydroxy-5-Hydroxymethyl-L-Proline]
Azetidine Iminosugars From The Cyclization Of 3,5-Di- O -Triflates Of Α-Furanosides And Of 2,4-Di- O -Triflates Of Β-Pyranosides Derived From Glucose
N-(2-Carboxyethyl)-2,5-Dideoxy-2,5-Imino-D-Mannonic Acid [(3r,4r,5r)-1-(2-Carboxyethyl)-3,4-Dihydroxy-5-Hydroxymethyl-L-Proline]
Glycosidase Inhibition By All 10 Stereoisomeric 2,5-Dideoxy-2,5- Iminohexitols Prepared From The Enantiomers Of Glucuronolactone
N-(2-Carboxyethyl)-2,5-Dideoxy-2,5-Imino-D-Mannonic Acid [(3r,4r,5r)-1-(2-Carboxyethyl)-3,4-Dihydroxy-5-Hydroxymethyl-L-Proline]
Glycosidase Inhibition By All 10 Stereoisomeric 2,5-Dideoxy-2,5- Iminohexitols Prepared From The Enantiomers Of Glucuronolactone
Synthesis From D-Altrose Of (5 R,6 R,7 R,8 S)-5,7-Dihydroxy-8- Hydroxymethylconidine And 2,4-Dideoxy-2,4-Imino-D-Glucitol, Azetidine Analogues Of Swainsonine And 1,4-Dideoxy-1,4-Imino-D-Mannitol
Glycosidase Inhibition By All 10 Stereoisomeric 2,5-Dideoxy-2,5- Iminohexitols Prepared From The Enantiomers Of Glucuronolactone
Synthesis From D-Altrose Of (5 R,6 R,7 R,8 S)-5,7-Dihydroxy-8- Hydroxymethylconidine And 2,4-Dideoxy-2,4-Imino-D-Glucitol, Azetidine Analogues Of Swainsonine And 1,4-Dideoxy-1,4-Imino-D-Mannitol
Tautomerism In Schiff Bases. The Cases Of 2-Hydroxy-1-Naphthaldehyde And 1-Hydroxy-2-Naphthaldehyde Investigated In Solution And The Solid State
Synthesis From D-Altrose Of (5 R,6 R,7 R,8 S)-5,7-Dihydroxy-8- Hydroxymethylconidine And 2,4-Dideoxy-2,4-Imino-D-Glucitol, Azetidine Analogues Of Swainsonine And 1,4-Dideoxy-1,4-Imino-D-Mannitol
Tautomerism In Schiff Bases. The Cases Of 2-Hydroxy-1-Naphthaldehyde And 1-Hydroxy-2-Naphthaldehyde Investigated In Solution And The Solid State
Schiff Bases From Tris And Ortho-Hydroxyarenecarbaldehydes: Structures And Tautomeric Equilibria In The Solid State And In Solution
Tautomerism In Schiff Bases. The Cases Of 2-Hydroxy-1-Naphthaldehyde And 1-Hydroxy-2-Naphthaldehyde Investigated In Solution And The Solid State
Schiff Bases From Tris And Ortho-Hydroxyarenecarbaldehydes: Structures And Tautomeric Equilibria In The Solid State And In Solution
A Quantitative Structure-Reactivity Relationship In N-Acetyl Oxazolidines: An Electrostatic Interaction Controls Rotamer Population
Schiff Bases From Tris And Ortho-Hydroxyarenecarbaldehydes: Structures And Tautomeric Equilibria In The Solid State And In Solution
A Quantitative Structure-Reactivity Relationship In N-Acetyl Oxazolidines: An Electrostatic Interaction Controls Rotamer Population
Hydrazones From Hydroxy Naphthaldehydes And N-Aminoheterocycles: Structure And Stereodynamics
A Quantitative Structure-Reactivity Relationship In N-Acetyl Oxazolidines: An Electrostatic Interaction Controls Rotamer Population
Hydrazones From Hydroxy Naphthaldehydes And N-Aminoheterocycles: Structure And Stereodynamics
Schiff Bases From Tris And Formylpyridines: Structure And Mechanistic Rationale Aided By Dft Calculations
Hydrazones From Hydroxy Naphthaldehydes And N-Aminoheterocycles: Structure And Stereodynamics
Schiff Bases From Tris And Formylpyridines: Structure And Mechanistic Rationale Aided By Dft Calculations
An Anomeric Effect Drives The Regiospecific Ring-Opening Of 1,3-Oxazolidines Under Acetylating Conditions
Schiff Bases From Tris And Formylpyridines: Structure And Mechanistic Rationale Aided By Dft Calculations
An Anomeric Effect Drives The Regiospecific Ring-Opening Of 1,3-Oxazolidines Under Acetylating Conditions
An Efficient And Highly Diastereoselective Synthesis Of C-Glycosylated 1,3-Oxazolidines From N-Methyl-D-Glucamine
An Anomeric Effect Drives The Regiospecific Ring-Opening Of 1,3-Oxazolidines Under Acetylating Conditions
An Efficient And Highly Diastereoselective Synthesis Of C-Glycosylated 1,3-Oxazolidines From N-Methyl-D-Glucamine
Catalytic Screening For 1,2-Diol Protection: A Saccharose-Derived Hydrothermal Carbon Showcases Enhanced Performance
WEB ACCESIBLE