PUBLICACIÓN

Nine of 16 stereoisomeric polyhydroxylated proline amides are potent β-N-acetylhexosaminidase inhibitors

ACCEDER A LA PUBLICACIÓN: Scopus Orcid

Ayers B.J. et al.

2014 JOURNAL OF ORGANIC CHEMISTRY

Organic Chemistry (Q1)

JCR: 4.721

SJR: 2.007

CITAS

31

DOI

10.1021/jo500157p

EID

2-s2.0-84898967445

ISSN

0022-3263

EISSN

1520-6904

AUTORES DE LA UEX

Rafael Fernando Martínez Vázquez

OTRAS PUBLICACIONES DE INTERÉS

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Tuning Synthesis And Sonochemistry Forges Learning And Enhances Educational Training: Protection Of 1,3-Diols Under Heterogeneous Catalysis As Sustainable Case Study
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Tuning Synthesis And Sonochemistry Forges Learning And Enhances Educational Training: Protection Of 1,3-Diols Under Heterogeneous Catalysis As Sustainable Case Study
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A True Reverse Anomeric Effect Does Exist After All: A Hydrogen Bonding Stereocontrolling Effect In 2-Iminoaldoses
Síntesis De Acetales Derivados De 1,2-Dioles En Presencia De Catalizadores Ácidos Carbonosos
A True Reverse Anomeric Effect Does Exist After All: A Hydrogen Bonding Stereocontrolling Effect In 2-Iminoaldoses
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Targeting The Ftsz Allosteric Binding Site With A Novel Fluorescence Polarization Screen, Cytological And Structural Approaches For Antibacterial Discovery
Organic Sonochemistry: A Chemist's Timely Perspective On Mechanisms And Reactivity
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A Novel Agonist Of The Type 1 Lysophosphatidic Acid Receptor (Lpa1), Ucm-05194, Shows Efficacy In Neuropathic Pain Amelioration
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Imine Or Enamine? Insights And Predictive Guidelines From The Electronic Effect Of Substituents In H-Bonded Salicylimines
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Isolation From Stevia Rebaudiana Of Dmdp Acetic Acid, A Novel Iminosugar Amino Acid: Synthesis And Glycosidase Inhibition Profile Of Glycine And Β-Alanine Pyrrolidine Amino Acids
Cycloadditions With Mesoionic Dipoles: Strategy And Control
Isolation From Stevia Rebaudiana Of Dmdp Acetic Acid, A Novel Iminosugar Amino Acid: Synthesis And Glycosidase Inhibition Profile Of Glycine And Β-Alanine Pyrrolidine Amino Acids
Cycloadditions With Mesoionic Dipoles: Strategy And Control
The Dimroth Rearrangement As A Probable Cause For Structural Misassignments In Imidazo[1,2-A]pyrimidines: A 15n-Labelling Study And An Easy Method For The Determination Of Regiochemistry
Cycloadditions With Mesoionic Dipoles: Strategy And Control
The Dimroth Rearrangement As A Probable Cause For Structural Misassignments In Imidazo[1,2-A]pyrimidines: A 15n-Labelling Study And An Easy Method For The Determination Of Regiochemistry
The Structural Assembly Switch Of Cell Division Protein Ftsz Probed With Fluorescent Allosteric Inhibitors
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The Structural Assembly Switch Of Cell Division Protein Ftsz Probed With Fluorescent Allosteric Inhibitors
Cycloadditions With Mesoionic Dipoles: Strategy And Control
The Structural Assembly Switch Of Cell Division Protein Ftsz Probed With Fluorescent Allosteric Inhibitors
Cycloadditions With Mesoionic Dipoles: Strategy And Control
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Short And Sweet: D-Glucose To L-Glucose And L-Glucuronic Acid
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Short And Sweet: D-Glucose To L-Glucose And L-Glucuronic Acid
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Kurz Und Knapp:l-Glucose Undl-Glucuronsäure Ausd-Glucose
Synthesis Of The Enantiomers Of Xylnac And Lyxnac: Comparison Of Β-N-Acetylhexosaminidase Inhibition By The 8 Stereoisomers Of 2-N-Acetylamino-1,2,4-Trideoxy-1,4-Iminopentitols
Kurz Und Knapp:l-Glucose Undl-Glucuronsäure Ausd-Glucose
Hydrazones From Hydroxy Naphthaldehydes. Part 2. Condensations With Aromatic N-Aminoheterocycles And Elucidation Of Tautomeric Structures
Kurz Und Knapp:l-Glucose Undl-Glucuronsäure Ausd-Glucose
Hydrazones From Hydroxy Naphthaldehydes. Part 2. Condensations With Aromatic N-Aminoheterocycles And Elucidation Of Tautomeric Structures
(3r,4s,5r,6r,7s)-3,4,5,7-Tetrahydroxyconidine, An Azetidine Analogue Of 6,7-Diepicastanospermine And A Conformationally Constrained D- Deoxyaltronojirimycin, From L-Arabinose
Hydrazones From Hydroxy Naphthaldehydes. Part 2. Condensations With Aromatic N-Aminoheterocycles And Elucidation Of Tautomeric Structures
(3r,4s,5r,6r,7s)-3,4,5,7-Tetrahydroxyconidine, An Azetidine Analogue Of 6,7-Diepicastanospermine And A Conformationally Constrained D- Deoxyaltronojirimycin, From L-Arabinose
C-Branched Iminosugars: Α-Glucosidase Inhibition By Enantiomers Of Isodmdp, Isodgdp, And Isodab- L -Isodmdp Compared To Miglitol And Miglustat
(3r,4s,5r,6r,7s)-3,4,5,7-Tetrahydroxyconidine, An Azetidine Analogue Of 6,7-Diepicastanospermine And A Conformationally Constrained D- Deoxyaltronojirimycin, From L-Arabinose
C-Branched Iminosugars: Α-Glucosidase Inhibition By Enantiomers Of Isodmdp, Isodgdp, And Isodab- L -Isodmdp Compared To Miglitol And Miglustat
Azetidine Iminosugars From The Cyclization Of 3,5-Di- O -Triflates Of Α-Furanosides And Of 2,4-Di- O -Triflates Of Β-Pyranosides Derived From Glucose
C-Branched Iminosugars: Α-Glucosidase Inhibition By Enantiomers Of Isodmdp, Isodgdp, And Isodab- L -Isodmdp Compared To Miglitol And Miglustat
Azetidine Iminosugars From The Cyclization Of 3,5-Di- O -Triflates Of Α-Furanosides And Of 2,4-Di- O -Triflates Of Β-Pyranosides Derived From Glucose
N-(2-Carboxyethyl)-2,5-Dideoxy-2,5-Imino-D-Mannonic Acid [(3r,4r,5r)-1-(2-Carboxyethyl)-3,4-Dihydroxy-5-Hydroxymethyl-L-Proline]
Azetidine Iminosugars From The Cyclization Of 3,5-Di- O -Triflates Of Α-Furanosides And Of 2,4-Di- O -Triflates Of Β-Pyranosides Derived From Glucose
N-(2-Carboxyethyl)-2,5-Dideoxy-2,5-Imino-D-Mannonic Acid [(3r,4r,5r)-1-(2-Carboxyethyl)-3,4-Dihydroxy-5-Hydroxymethyl-L-Proline]
Glycosidase Inhibition By All 10 Stereoisomeric 2,5-Dideoxy-2,5- Iminohexitols Prepared From The Enantiomers Of Glucuronolactone
N-(2-Carboxyethyl)-2,5-Dideoxy-2,5-Imino-D-Mannonic Acid [(3r,4r,5r)-1-(2-Carboxyethyl)-3,4-Dihydroxy-5-Hydroxymethyl-L-Proline]
Glycosidase Inhibition By All 10 Stereoisomeric 2,5-Dideoxy-2,5- Iminohexitols Prepared From The Enantiomers Of Glucuronolactone
Synthesis From D-Altrose Of (5 R,6 R,7 R,8 S)-5,7-Dihydroxy-8- Hydroxymethylconidine And 2,4-Dideoxy-2,4-Imino-D-Glucitol, Azetidine Analogues Of Swainsonine And 1,4-Dideoxy-1,4-Imino-D-Mannitol
Glycosidase Inhibition By All 10 Stereoisomeric 2,5-Dideoxy-2,5- Iminohexitols Prepared From The Enantiomers Of Glucuronolactone
Synthesis From D-Altrose Of (5 R,6 R,7 R,8 S)-5,7-Dihydroxy-8- Hydroxymethylconidine And 2,4-Dideoxy-2,4-Imino-D-Glucitol, Azetidine Analogues Of Swainsonine And 1,4-Dideoxy-1,4-Imino-D-Mannitol
Tautomerism In Schiff Bases. The Cases Of 2-Hydroxy-1-Naphthaldehyde And 1-Hydroxy-2-Naphthaldehyde Investigated In Solution And The Solid State
Synthesis From D-Altrose Of (5 R,6 R,7 R,8 S)-5,7-Dihydroxy-8- Hydroxymethylconidine And 2,4-Dideoxy-2,4-Imino-D-Glucitol, Azetidine Analogues Of Swainsonine And 1,4-Dideoxy-1,4-Imino-D-Mannitol
Tautomerism In Schiff Bases. The Cases Of 2-Hydroxy-1-Naphthaldehyde And 1-Hydroxy-2-Naphthaldehyde Investigated In Solution And The Solid State
Schiff Bases From Tris And Ortho-Hydroxyarenecarbaldehydes: Structures And Tautomeric Equilibria In The Solid State And In Solution
Tautomerism In Schiff Bases. The Cases Of 2-Hydroxy-1-Naphthaldehyde And 1-Hydroxy-2-Naphthaldehyde Investigated In Solution And The Solid State
Schiff Bases From Tris And Ortho-Hydroxyarenecarbaldehydes: Structures And Tautomeric Equilibria In The Solid State And In Solution
A Quantitative Structure-Reactivity Relationship In N-Acetyl Oxazolidines: An Electrostatic Interaction Controls Rotamer Population
Schiff Bases From Tris And Ortho-Hydroxyarenecarbaldehydes: Structures And Tautomeric Equilibria In The Solid State And In Solution
A Quantitative Structure-Reactivity Relationship In N-Acetyl Oxazolidines: An Electrostatic Interaction Controls Rotamer Population
Hydrazones From Hydroxy Naphthaldehydes And N-Aminoheterocycles: Structure And Stereodynamics
A Quantitative Structure-Reactivity Relationship In N-Acetyl Oxazolidines: An Electrostatic Interaction Controls Rotamer Population
Hydrazones From Hydroxy Naphthaldehydes And N-Aminoheterocycles: Structure And Stereodynamics
Schiff Bases From Tris And Formylpyridines: Structure And Mechanistic Rationale Aided By Dft Calculations
Hydrazones From Hydroxy Naphthaldehydes And N-Aminoheterocycles: Structure And Stereodynamics
Schiff Bases From Tris And Formylpyridines: Structure And Mechanistic Rationale Aided By Dft Calculations
An Anomeric Effect Drives The Regiospecific Ring-Opening Of 1,3-Oxazolidines Under Acetylating Conditions
Schiff Bases From Tris And Formylpyridines: Structure And Mechanistic Rationale Aided By Dft Calculations
An Anomeric Effect Drives The Regiospecific Ring-Opening Of 1,3-Oxazolidines Under Acetylating Conditions
An Efficient And Highly Diastereoselective Synthesis Of C-Glycosylated 1,3-Oxazolidines From N-Methyl-D-Glucamine
An Anomeric Effect Drives The Regiospecific Ring-Opening Of 1,3-Oxazolidines Under Acetylating Conditions
An Efficient And Highly Diastereoselective Synthesis Of C-Glycosylated 1,3-Oxazolidines From N-Methyl-D-Glucamine
Catalytic Screening For 1,2-Diol Protection: A Saccharose-Derived Hydrothermal Carbon Showcases Enhanced Performance
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