PUBLICACIÓN

Synthesis of the enantiomers of XYLNAc and LYXNAc: Comparison of β-N-acetylhexosaminidase inhibition by the 8 stereoisomers of 2-N-acetylamino-1,2,4-trideoxy-1,4-iminopentitols

ACCEDER A LA PUBLICACIÓN: Scopus Orcid

2014 Organic and Biomolecular Chemistry

Biochemistry (Q1), Organic Chemistry (Q1), Physical and Theoretical Chemistry (Q1)

JCR: 3.562

SJR: 1.396

CITAS

19

DOI

10.1039/c4ob00097h

EID

2-s2.0-84901251361

ISSN

1477-0520

BIBTEX

@article{Crabtree_2014, doi = {10.1039/c4ob00097h}, url = {https://doi.org/10.1039%2Fc4ob00097h}, year = 2014, publisher = {Royal Society of Chemistry ({RSC})}, volume = {12}, number = {23}, pages = {3932}, author = {Elizabeth V. Crabtree and R. Fernando Mart{\'{\i}}nez and Shinpei Nakagawa and Isao Adachi and Terry D. Butters and Atsushi Kato and George W. J. Fleet and Andreas F. G. Glawar}, title = {Synthesis of the enantiomers of {XYLNAc} and {LYXNAc}: comparison of $\upbeta$-N-acetylhexosaminidase inhibition by the 8 stereoisomers of 2-N-acetylamino-1,2,4-trideoxy-1,4-iminopentitols}, journal = {Organic {\&} Biomolecular Chemistry}}

AUTORES DE LA UEX

Rafael Fernando Martínez Vázquez

OTRAS PUBLICACIONES DE INTERÉS

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Short And Sweet: D-Glucose To L-Glucose And L-Glucuronic Acid
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Kurz Und Knapp:l-Glucose Undl-Glucuronsäure Ausd-Glucose
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Hydrazones From Hydroxy Naphthaldehydes. Part 2. Condensations With Aromatic N-Aminoheterocycles And Elucidation Of Tautomeric Structures
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Hydrazones From Hydroxy Naphthaldehydes. Part 2. Condensations With Aromatic N-Aminoheterocycles And Elucidation Of Tautomeric Structures
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Hydrazones From Hydroxy Naphthaldehydes. Part 2. Condensations With Aromatic N-Aminoheterocycles And Elucidation Of Tautomeric Structures
(3r,4s,5r,6r,7s)-3,4,5,7-Tetrahydroxyconidine, An Azetidine Analogue Of 6,7-Diepicastanospermine And A Conformationally Constrained D- Deoxyaltronojirimycin, From L-Arabinose
C-Branched Iminosugars: Α-Glucosidase Inhibition By Enantiomers Of Isodmdp, Isodgdp, And Isodab- L -Isodmdp Compared To Miglitol And Miglustat
(3r,4s,5r,6r,7s)-3,4,5,7-Tetrahydroxyconidine, An Azetidine Analogue Of 6,7-Diepicastanospermine And A Conformationally Constrained D- Deoxyaltronojirimycin, From L-Arabinose
C-Branched Iminosugars: Α-Glucosidase Inhibition By Enantiomers Of Isodmdp, Isodgdp, And Isodab- L -Isodmdp Compared To Miglitol And Miglustat
Azetidine Iminosugars From The Cyclization Of 3,5-Di- O -Triflates Of Α-Furanosides And Of 2,4-Di- O -Triflates Of Β-Pyranosides Derived From Glucose
C-Branched Iminosugars: Α-Glucosidase Inhibition By Enantiomers Of Isodmdp, Isodgdp, And Isodab- L -Isodmdp Compared To Miglitol And Miglustat
Azetidine Iminosugars From The Cyclization Of 3,5-Di- O -Triflates Of Α-Furanosides And Of 2,4-Di- O -Triflates Of Β-Pyranosides Derived From Glucose
N-(2-Carboxyethyl)-2,5-Dideoxy-2,5-Imino-D-Mannonic Acid [(3r,4r,5r)-1-(2-Carboxyethyl)-3,4-Dihydroxy-5-Hydroxymethyl-L-Proline]
Azetidine Iminosugars From The Cyclization Of 3,5-Di- O -Triflates Of Α-Furanosides And Of 2,4-Di- O -Triflates Of Β-Pyranosides Derived From Glucose
N-(2-Carboxyethyl)-2,5-Dideoxy-2,5-Imino-D-Mannonic Acid [(3r,4r,5r)-1-(2-Carboxyethyl)-3,4-Dihydroxy-5-Hydroxymethyl-L-Proline]
Glycosidase Inhibition By All 10 Stereoisomeric 2,5-Dideoxy-2,5- Iminohexitols Prepared From The Enantiomers Of Glucuronolactone
N-(2-Carboxyethyl)-2,5-Dideoxy-2,5-Imino-D-Mannonic Acid [(3r,4r,5r)-1-(2-Carboxyethyl)-3,4-Dihydroxy-5-Hydroxymethyl-L-Proline]
Glycosidase Inhibition By All 10 Stereoisomeric 2,5-Dideoxy-2,5- Iminohexitols Prepared From The Enantiomers Of Glucuronolactone
Synthesis From D-Altrose Of (5 R,6 R,7 R,8 S)-5,7-Dihydroxy-8- Hydroxymethylconidine And 2,4-Dideoxy-2,4-Imino-D-Glucitol, Azetidine Analogues Of Swainsonine And 1,4-Dideoxy-1,4-Imino-D-Mannitol
Glycosidase Inhibition By All 10 Stereoisomeric 2,5-Dideoxy-2,5- Iminohexitols Prepared From The Enantiomers Of Glucuronolactone
Synthesis From D-Altrose Of (5 R,6 R,7 R,8 S)-5,7-Dihydroxy-8- Hydroxymethylconidine And 2,4-Dideoxy-2,4-Imino-D-Glucitol, Azetidine Analogues Of Swainsonine And 1,4-Dideoxy-1,4-Imino-D-Mannitol
Tautomerism In Schiff Bases. The Cases Of 2-Hydroxy-1-Naphthaldehyde And 1-Hydroxy-2-Naphthaldehyde Investigated In Solution And The Solid State
Synthesis From D-Altrose Of (5 R,6 R,7 R,8 S)-5,7-Dihydroxy-8- Hydroxymethylconidine And 2,4-Dideoxy-2,4-Imino-D-Glucitol, Azetidine Analogues Of Swainsonine And 1,4-Dideoxy-1,4-Imino-D-Mannitol
Tautomerism In Schiff Bases. The Cases Of 2-Hydroxy-1-Naphthaldehyde And 1-Hydroxy-2-Naphthaldehyde Investigated In Solution And The Solid State
Schiff Bases From Tris And Ortho-Hydroxyarenecarbaldehydes: Structures And Tautomeric Equilibria In The Solid State And In Solution
Tautomerism In Schiff Bases. The Cases Of 2-Hydroxy-1-Naphthaldehyde And 1-Hydroxy-2-Naphthaldehyde Investigated In Solution And The Solid State
Schiff Bases From Tris And Ortho-Hydroxyarenecarbaldehydes: Structures And Tautomeric Equilibria In The Solid State And In Solution
A Quantitative Structure-Reactivity Relationship In N-Acetyl Oxazolidines: An Electrostatic Interaction Controls Rotamer Population
Schiff Bases From Tris And Ortho-Hydroxyarenecarbaldehydes: Structures And Tautomeric Equilibria In The Solid State And In Solution
A Quantitative Structure-Reactivity Relationship In N-Acetyl Oxazolidines: An Electrostatic Interaction Controls Rotamer Population
Hydrazones From Hydroxy Naphthaldehydes And N-Aminoheterocycles: Structure And Stereodynamics
A Quantitative Structure-Reactivity Relationship In N-Acetyl Oxazolidines: An Electrostatic Interaction Controls Rotamer Population
Hydrazones From Hydroxy Naphthaldehydes And N-Aminoheterocycles: Structure And Stereodynamics
Schiff Bases From Tris And Formylpyridines: Structure And Mechanistic Rationale Aided By Dft Calculations
Hydrazones From Hydroxy Naphthaldehydes And N-Aminoheterocycles: Structure And Stereodynamics
Schiff Bases From Tris And Formylpyridines: Structure And Mechanistic Rationale Aided By Dft Calculations
An Anomeric Effect Drives The Regiospecific Ring-Opening Of 1,3-Oxazolidines Under Acetylating Conditions
Schiff Bases From Tris And Formylpyridines: Structure And Mechanistic Rationale Aided By Dft Calculations
An Anomeric Effect Drives The Regiospecific Ring-Opening Of 1,3-Oxazolidines Under Acetylating Conditions
An Efficient And Highly Diastereoselective Synthesis Of C-Glycosylated 1,3-Oxazolidines From N-Methyl-D-Glucamine
An Anomeric Effect Drives The Regiospecific Ring-Opening Of 1,3-Oxazolidines Under Acetylating Conditions
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